试题与答案

下列对吩噻嗪类抗精神药构效关系的叙述不正确的是() A.2位被吸电子基团取代时活性增

题型:单项选择题 A1/A2型题

题目:

下列对吩噻嗪类抗精神药构效关系的叙述不正确的是()

A.2位被吸电子基团取代时活性增强

B.吩噻嗪10位氮原子与侧链碱性氨基氮原子间相隔2个碳原子为宜

C.侧链上碱性氨基,可以是二甲氨基或哌嗪基等

D.吩噻嗪环10位氮原子换成碳原子,再通过双键与侧链相连接,为噻吨类抗精神病药

E.碱性侧链末端含伯醇基时,可制成长链脂肪酸酯的前药,可使作用时间延长

答案:

参考答案:B

解析:以上对吩噻嗪类抗精神药构效关系正确的是2位被吸电子基团取代时活性增强。吩噻嗪10位氮原子与侧链碱性氨基氮原子间相隔3个碳原子为宜。侧链上碱性氨基,可以是二甲氨基或哌嗪基等。吩噻嗪环10位氮原子换成碳原子,再通过双键与侧链相连接,为噻吨类抗精神病药。碱性侧链末端含伯醇基时,可制成长链脂肪酸酯的前药,可使作用时间延长。所以答案为B。

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题型:阅读理解

  Microwaves may be great at warming up food, but what about warming people?

Using microwaves to directly heat owners of a room would save much of the energy wasted by heating walls and furniture. And despite popular ideas about microwaves, this technique would be safe, according to Charles R. Buffler of the Microwave Research Center in Marlborough, New Hampshire. Low-power microwaves only penetrate (贯穿) the skin (low-power microwave penetration in a ham is about 0.2 inches, for example) and with no negative effects.

To test this idea, Buffler subjected himself to microwaves in a special room using a standard 500-watt, 2459 MHz magnetron (磁控管). He found that a person will start to feel warmth at about 20 milliwatts per square centimeter (mw. /sq.cm.); a satisfactory feeling of warmth occurs between 35 and 50 mw./sq.cm. By comparison, a person standing in noonday summer sun feels the amount of 85 mw./sq.cm. And a frozen meat pie in your microwave oven receives about 1000 mw./sq. cm.

In houses of the future, each room could be provided with its own magnetron, says Buffler. When you stepped into the living room, for example, a motion detector would turn on the magnetron, filling the room with low-power microwaves. In the same way that a microwaves oven heats up a hamburger, but not the plate it’s on, you would feel warmth from the microwaves without changing the temperature of your coffee table. (You could, however, make your favorite easy chair even more comfortable by treating it with a radiation-absorbing chemical.)

While it might be some time before homeowners are comfortable enough with the idea to set up whole body microwave heaters in houses, Buffler says microwaves may attract livestock farmers. Lambs that are born outdoors in winter, for example, are frequently lost to cold. Microwaves could warm the lambs safely and quickly.

小题1: Which of the following can tell the main idea of the passage?

A.A new heating system.

B.A new microwave oven.

C.A popular technique.

D.The magnetron.小题2: The test conducted by Buffler shows that when a person feels comfortable warmth, he receives about ____.

A.20 mw. / sq. cm.

B.40 mw. / sq. cm.

C.60 mw. / sq. cm.

D.85 mw. / sq. cm.小题3: According to paragraph 4, which of the following fills the room with low-power microwaves?

A.The magnetron.

B.The motion detector.

C.The microwave oven.

D.The radiation-absorbing chemical.小题4: Which of the following statements about microwave heaters would Buffler most probably agree with?

A.Microwave heaters will soon be widely used by homeowners.

B.Microwave heaters sometimes make people feel uncomfortable.

C.Microwave heaters will be probably first used by livestock farmers to protect their lambs in winter.

D.Microwave heaters cannot be accepted by the public because they are somewhat unsafe.

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